3-Bromocytisine

3-Bromocytisine (3-Br-cytisine) is a potent nACh receptors agonist, with IC50s are 0.28, 0.30 and 31.6 nM for hα4β4, hα4β2, and hα7-nACh, respectively. 3-Bromocytisine (3-Br-cytisine) shows different effects on high (HS) and low (LS) ACh sensitivity α4β2 nAChRs with EC50s are 8 and 50 nM, respectively[1][2].


Cat. No.: EX-A14476	Purity: >98%

	Chemical structure of 3-Bromocytisine

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
50mg	575	In-stock
100mg	825	In-stock
250mg	1280	In-stock
500mg	1792	In-stock
1g	2508	In-stock

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Synonyms	3-Br-cytisine
CAS No.	207390-14-5
Purity	>98%
Formula	C11H13BrN2O
Mol Weight	269.138
Color	White to off-white
State	Solid
Solubility	soluble in DMSO
Shelf Life	>3 years if stored properly
Storage	Powder -20℃, 3 years; In solvent -20℃, 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Houlihan LM, et al. Activity of cytisine and its brominated isosteres on recombinant human alpha7, alpha4beta2 and alpha4beta4 nicotinic acetylcholine receptors. J Neurochem. 2001 Sep;78(5):1029-43. [2]. Moroni M, et al. alpha4beta2 nicotinic receptors with high and low acetylcholine sensitivity: pharmacology, stoichiometry, and sensitivity to long-term exposure to nicotine. Mol Pharmacol. 2006 Aug;70(2):755-68.
CoA	CoA of 3-Bromocytisine

Smiles:	C1[C@H]2CNC[C@@H]1C3=CC=C(C(=O)N3C2)Br


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