SCH-772984

SCH772984 is a novel, specific inhibitor of ERK1/2 with IC50 values of 4 nM and 1 nM in cell-free assay, respectively, And show robust efficacy in RAS- or BRAF-mutant cancer cells.


Cat. No.: EX-A296	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock	Quantity	Order
500mg	2000	In-stock

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CAS No.	942183-80-4
Purity	>98%
Formula	C33H33N9O2
Mol Weight	587.6742
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Morris EJ, et al. Discovery of a novel ERK inhibitor with activity in models of acquired resistance to BRAF and MEK inhibitors. Cancer Discov, 2013 Apr 29.
CoA	CoA of SCH-772984

Smiles:	O=C(CN1CC[C@H](C1)C(=O)NC1=CC2=C(NN=C2C2=CC=NC=C2)C=C1)N1CCN(CC1)C1=CC=C(C=C1)C1=NC=CC=N1


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