S1RA

S1RA is a selective sigma-1 receptor antagonist, with a reported binding affinity of Ki = 17.0 ± 7.0 nM, selective over the sigma-2 receptor and against a panel of other 170 receptors, enzymes, transporters and ion channels.


Cat. No.: EX-A357	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	480	In-stock
250mg	690	In-stock
500mg	890	In-stock
1g	1650	In-stock
5g	6600	In-stock
10g	10560	In-stock

Send PO to E-mail:order@excenen.com; or Fax:+86 020 81619670

Discount Request


Synonyms	E-52862 HCl
CAS No.	878141-96-9
Purity	>98%
Formula	C20H24ClN3O2
Mol Weight	373.876
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. L Romero, et al. Pharmacological properties of S1RA, a new sigma-1 receptor antagonist that inhibits neuropathic pain and activity-induced spinal sensitization. Br J Pharmacol. 2012, 166(8): 2289–2306.
CoA	CoA of S1RA

Smiles:	Cl.CC1=CC(OCCN2CCOCC2)=NN1C1=CC2=CC=CC=C2C=C1


		Search