Tariquidar

Tariquidar (XR9576) is a potent and selective noncompetitive inhibitor of P-glycoprotein with Kd of 5.1 nM in CHrB30 cell line, reverses drug resistance in MDR cell Lines.


Cat. No.: EX-A231	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	350	In-stock
200mg	550	In-stock
500mg	785	In-stock
1g	1085	In-stock
5g	3500	In-stock

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Synonyms	XR9576
CAS No.	206873-63-4
Purity	>98%
Formula	C38H38N4O6
Mol Weight	646.7315
Appearance	Solid powder
Solubility	Soluble in DMSO, not in water
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Martin C, et al. The molecular interaction of the high affinity reversal agent XR9576 with P-glycoprotein. Br J Pharmacol, 1999, 128(2), 403-411. [2]. Mistry P, et al. In vitro and in vivo reversal of P-glycoprotein-mediated multidrug resistance by a novel potent modulator, XR9576. Cancer Res, 2001, 61(2), 749-758. [3]. Robey, Robert W et al. “Pheophorbide a is a specific probe for ABCG2 function and inhibition.” Cancer research vol. 64,4 (2004): 1242-6.
CoA	CoA of Tariquidar

Smiles:	COC1=CC2=C(CN(CCC3=CC=C(NC(=O)C4=CC(OC)=C(OC)C=C4NC(=O)C4=CC5=CC=CC=C5N=C4)C=C3)CC2)C=C1OC


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