R-GNE-140

(R)-GNE-140 is a potent lactate dehydrogenase A (LDHA) inhibitor, with IC50s of 3 nM and 5 nM for LDHA and LDHB, respectively; (R)-GNE-140 is 18-fold more potent than S enantiomer.


Cat. No.: EX-A1474	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	800	In-stock
500mg	1200	In-stock
1g	1685	In-stock
2g	2696	In-stock
5g	5500	In-stock
10g	8600	In-stock

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Synonyms	(R)-GNE-140
CAS No.	2003234-63-5
Purity	>98%
Formula	C25H23ClN2O3S2
Mol Weight	499.045
Appearance	Solid powder
Solubility	soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Purkey HE, et al. Cell Active Hydroxylactam Inhibitors of Human Lactate Dehydrogenase with Oral Bioavailability in Mice. ACS Med Chem Lett. 2016 Aug 26;7(10):896-901.
CoA	CoA of R-GNE-140

Smiles:	OC1=C(SC2=CC=CC=C2Cl)C(=O)N[C@@](C1)(C1=CSC=C1)C1=CC=C(C=C1)N1CCOCC1


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