GSK6853

GSK6853 is a potent and selective inhibitor of the BRPF1 bromodomain. GSK6853 shows excellent BRPF1 potency (pKd=9.5) and greater than 1600-fold selectivity over all other bromodomains.


Cat. No.: EX-A1080	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
250mg	550	In-stock
500mg	800	In-stock
1g	1300	In-stock
5g	4450	In-stock
10g	6880	In-stock

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CAS No.	1910124-24-1
Purity	>98%
Formula	C22H27N5O3
Mol Weight	409.4815
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Bamborough P et al. GSK6853, a Chemical Probe for Inhibition of the BRPF1 Bromodomain. ACS Med Chem Lett. 2016 May 9;7(6):552-7.
CoA	CoA of GSK6853

Smiles:	COC1=CC=CC=C1C(=O)NC1=C(C=C2N(C)C(=O)N(C)C2=C1)N1CCNC[C@H]1C


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