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Product Information:

THZ531

THZ531 is a selective and covalent inhibitor of both CDK12 and CDK13 with IC50s of 158 nM and 69 nM, respectively.

Cat. No.: EX-A1532    Purity: >98%
THZ531
For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
50mg425In-stock
100mg650In-stock
250mg850In-stock
500mg1150In-stock
1g1650In-stock
5g4850In-stock


CAS No.1702809-17-3
Purity>98%
FormulaC30H32ClN7O2
Mol Weight558.074
Appearancesolid powder
SolubilitySoluble in DMSO
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Zhang T, et al. Covalent targeting of remote cysteine residues to develop CDK12 and CDK13 inhibitors. Nat Chem Biol. 2016 Oct;12(10):876-84.

CoACoA of THZ531
Smiles:CN(C)C\C=C\C(=O)NC1=CC=C(C=C1)C(=O)N1CCC[C@H](C1)NC1=NC(C2=CNC3=C2C=CC=C3)=C(Cl)C=N1

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