ARQ-092

Miransertib (ARQ-092) is an orally bioavailable, selective, and potent allosteric Akt inhibitor with IC50s of 2.7 nM, 14 nM and 8.1 nM for Akt1, Akt2, Akt3, respectively.


Cat. No.: EX-A1268	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	690	In-stock
250mg	1200	In-stock
500mg	1750	In-stock
1g	2600	In-stock

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Synonyms	Miransertib
CAS No.	1313881-70-7
Purity	>98%
Formula	C27H24N6
Mol Weight	432.5197
Appearance	Solid powder
Solubility	DMSO > 10mg/mL
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Lapierre JM, et al. Discovery of 3-(3-(4-(1-Aminocyclobutyl)phenyl)-5-phenyl-3H-imidazo[4,5-b]pyridin-2-yl)pyridin-2-amine (ARQ 092): An Orally Bioavailable, Selective, and Potent Allosteric AKT Inhibitor. J Med Chem. 2016 Jul 14;59(13):6455-69.
CoA	CoA of ARQ-092

Smiles:	NC1=NC=CC=C1C1=NC2=CC=C(N=C2N1C1=CC=C(C=C1)C1(N)CCC1)C1=CC=CC=C1


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