BI-3802

BI-3802 is a highly potent oncogenic transcription factor BCL6 degrader with strong de-repression of target genes anti-proliferative effects. BI-3802 inhibits the BTB domain of BCL6 with IC50 of ≤3 nM. BI-3802 exhibits antitumor activity.


Cat. No.: EX-A3703	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
25mg	800	In-stock
50mg	1250	In-stock
100mg	2200	In-stock
200mg	get quote	In-stock
500mg	get quote	In-stock
1g	get quote	In-stock

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CAS No.	2166387-65-9
Purity	>98%
Formula	C24H29ClN6O3
Mol Weight	484.978
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. Kerres N, et al. Chemically Induced Degradation of the Oncogenic Transcription Factor BCL6. Cell Rep. 2017 Sep 19;20(12):2860-2875. [2]. Mikołaj Słabicki, et al. Small-molecule-induced polymerization triggers degradation of BCL6. Nature. 2020 Nov 18.
CoA	CoA of BI-3802

Smiles:	ClC1=CN=C(N2C[C@H](C)C[C@H](C)C2)N=C1NC3=CC(C=C(OCC(NC)=O)C(N4C)=O)=C4C=C3


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