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Product Information:

BMS-986195

Branebrutinib (BMS-986195) is a highly potent, selective covalent, irreversible inhibitor of Bruton’s tyrosine kinase (BTK), with an IC50 of 0.1 nM.

Cat. No.: EX-A2720    Purity: >98%
BMS-986195
For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
100mg500In-stock
250mg785In-stock
500mg1085In-stock
1g1585In-stock
2g2700In-stock
5g4850In-stock


SynonymsBranebrutinib
CAS No.1912445-55-6
Purity>98%
FormulaC20H23FN4O2
Mol Weight370.4206
Appearancesolid powder
SolubilityDMSO : >50 mg/mL (400 mM)
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Watterson, Scott H et al. Discovery of Branebrutinib (BMS-986195): A Strategy for Identifying a Highly Potent and Selective Covalent Inhibitor Providing Rapid in Vivo Inactivation of Bruton's Tyrosine Kinase (BTK). Journal of medicinal chemistry vol. 62,7 (2019): 3228-3250.

CoACoA of BMS-986195
Smiles:CC#CC(=O)N[C@H]1CCCN(C1)C1=C(F)C=C(C(N)=O)C2=C1C(C)=C(C)N2

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