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Product Information:

CPI-169

CPI-169 is a potent, and selective EZH2 inhibitor with IC50 of 0.24 nM, 0.51 nM, and 6.1 nM for EZH2 WT, EZH2 Y641N, and EZH1, respectively.

Cat. No.: EX-A1684    Purity: >98%
CPI-169
For research only, Do not use for Human!

SizeUnit Price (US$)StockQuantityOrder
100mg825In-stock
200mg1385In-stock
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5gget quote
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SynonymsCPI-169 R-enantiomer
CAS No.1802175-07-0
Purity>98%
FormulaC27H36N4O5S
Mol Weight528.664
Appearancesolid powder
SolubilitySoluble in DMSO
Shelf Life>2 years if stored properly
StoragePowder -20℃ 2 years; In solvent -20℃ 1 month;
ShippingShipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.
 
 
Reference:  

[1]. Bradley, William D et al. “EZH2 inhibitor efficacy in non-Hodgkin's lymphoma does not require suppression of H3K27 monomethylation.” Chemistry & biology vol. 21,11 (2014): 1463-75.

CoACoA of CPI-169
Smiles:CCS(=O)(=O)N1CCC(CC1)[C@@H](C)N1C(C)=C(C(=O)NCC2=C(OC)C=C(C)NC2=O)C2=C1C=CC=C2

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