CCT251236

CCT251236 is a highly potent, orally bioavailable inhibitor of the HSF1 stress pathway. Moreover, CCT251236 displayed efficacy in a human ovarian carcinoma xenograft model.


Cat. No.: EX-A1634	Purity: >98%

For research only, Do not use for Human!

Size	Unit Price (US$)	Stock
100mg	550	In-stock
200mg	900	In-stock
500mg	1285	In-stock
1g	1800	In-stock
5g	6000	Inquire

Send PO to E-mail:order@excenen.com; or Fax:+86 020 81619670

Discount Request


CAS No.	1693731-40-6
Purity	>98%
Formula	C32H32N4O5
Mol Weight	552.6203
Appearance	solid powder
Solubility	Soluble in DMSO
Shelf Life	>2 years if stored properly
Storage	Powder -20℃ 2 years; In solvent -20℃ 1 month;
Shipping	Shipped under ambient temperature as non-hazardous chemical. This product is stable enough for a few weeks during ordinary shipping and time spent in Customs.

Reference:	[1]. MD Cheeseman, et al. Discovery of a Chemical Probe Bisamide (CCT251236): An Orally Bioavailable Efficacious Pirin Ligand from a Heat Shock Transcription Factor 1 (HSF1) Phenotypic Screen. J Med Chem. 2017 Jan 12;60(1):180-201.
CoA	CoA of CCT251236

Smiles:	CC1=CC=C(NC(=O)C2=CC3=C(OCCO3)C=C2)C=C1NC(=O)C1=CC=C2N=C(OCCN3CCCC3)C=CC2=C1


		Search